By Clemens Lamberth, J?rgen Dinges

The chemistry of heterocycles is a vital department of natural chemistry. this can be on account that plenty of traditional products,
e. g. hormones, antibiotics, supplements, and so forth. are composed of heterocyclic buildings. usually, those compounds exhibit gains and are
for that reason utilized as prescribed drugs to regard illnesses or as pesticides, herbicides or fungicides in crop safety. This quantity offers very important agrochemicals. all of the 21 chapters covers in a concise demeanour one classification of heterocycles, truly dependent as follows:

* Structural formulation of most vital examples (market products)
*Short historical past of historical past or discovery
* usual syntheses of significant examples
* Mode of action
* attribute organic activity
* Structure-activity relationship
* extra chemistry details (e.g. extra modifications, replacement syntheses, metabolic pathways, etc.)
* References

A worthwhile one-stop reference resource for researchers in academia and in addition to for graduate scholars with profession aspirations in the
agrochemical chemistry.Content:
Chapter 1 the importance of Heterocycles for prescribed drugs and Agrochemicals* (pages 1–20): Dr. Clemens Lamberth and Dr. Jurgen Dinges
Chapter 2 Triazine Herbicides (pages 21–38): Andrew J. F. Edmunds
Chapter three Pyrimidinyl and Triazinylsulfonylurea Herbicides (pages 39–50): Mary Ann Hanagan and Atul Puri
Chapter four Acetohydroxyacid Synthase Inhibiting Triazolopyrimidine Herbicides (pages 51–60): Timothy C. Johnson, Richard okay. Mann, Paul R. Schmitzer and Roger E. Gast
Chapter five HPPD?Inhibiting Benzoylpyrazole Herbicides (pages 61–68): Matthias Witschel
Chapter 6 Pyridyloxyphenoxypropionate Herbicides: Inhibitors of Acetyl?CoA Carboxylase (pages 69–82): William G. Whittingham
Chapter 7 Imidazolinone Herbicides (pages 83–89): Dale Shaner
Chapter eight Protoporphyrinogen?IX?Oxidase?Inhibiting Uracil Herbicides (pages 91–101): George Theodoridis
Chapter nine Benzimidazole Fungicides (pages 103–118): Laura Quaranta
Chapter 10 Morpholine Fungicides for the remedy of Powdery mold (pages 119–127): Dr. Clemens Lamberth
Chapter eleven Sterol Biosynthesis Inhibiting Triazole Fungicides (pages 129–145): Paul Worthington
Chapter 12 Methionine Biosynthesis?Inhibiting Anilinopyrimidine Fungicides (pages 147–154): Clemens Lamberth
Chapter thirteen Phenylpyrrole Fungicides (pages 155–162): Dr. Clemens Lamberth
Chapter 14 Broad?Spectrum Fungicidally energetic Pyrimidinyldioxy Strobilurins Inhibiting the breathing Chain (pages 163–174): Dr. Clemens Lamberth
Chapter 15 Pyrazole Carboxamide Fungicides Inhibiting Succinate Dehydrogenase (pages 175–193): Harald Walter
Chapter sixteen Avermectin pesticides and Acaricides (pages 195–207): Thomas Pitterna
Chapter 17 Pyridine and Thiazole?Containing pesticides as powerful Agonists on Insect Nicotinic Acetylcholine Receptors (pages 209–223): Peter Jeschke
Chapter 18 Pyrazole and Pyrimidine Acaricides and pesticides appearing as Inhibitors of Mitochondrial Electron shipping at advanced I (pages 225–237): Ottmar Franz Huter
Chapter 19 Phenylpyrazole?Containing Fiprole pesticides (pages 239–250): Stefan Schnatterer
Chapter 20 Pyrazolylpyridine Activators of the Insect Ryanodine Receptor (pages 251–263): George P. Lahm, Thomas P. Selby, Thomas M. Stevenson, Daniel Cordova, I. Billy Annan and John T. Andaloro
Chapter 21 Tetronic Acid pesticides and Acaricides Inhibiting Acetyl?CoA Carboxylase (pages 265–278): Thomas Bretschneider, Reiner Fischer and Ralf Nauen

Show description

Read Online or Download Bioactive Heterocyclic Compound Classes: Agrochemicals PDF

Similar pharmacy books

Pharmacometrics: The Science of Quantitative Pharmacology

Pharmacometrics is the technological know-how of reading and describing pharmacology in a quantitative model. The pharmaceutical is integrating pharmacometrics into its drug improvement software, yet there's a loss of and want for skilled pharmacometricians due to the fact that fewer and less educational courses exist to coach them.

Enhancement in Drug Delivery

Enhancement in Drug Delivery
I learn this publication with nice curiosity and located that it includes very beneficial info. using enhancers is usually crucial within the layout of novel pharmaceutical items and new treatments. i feel that this e-book provides a concise, readable, and in-depth overview of the basics, functions, and optimizations of a few of the skill to advertise drug absorption for the main used management routes. The booklet comprises a variety of examples of particular supply platforms in addition to equipment in their overview either in vitro and in vivo. The reader is galvanized with new principles to decide on the right enhancer for a brand new product and is supplied with "pro" and "contra" concerning the use of particular permeation enhancement techniques.

The individuals are renowned foreign specialists from academia and undefined.

In end, this quantity presents a multidisciplinary and entire reference that could be successfully utilized by researchers within the pharmaceutical and academia in addition to a textbook for pharmacy scholars at a number of degrees. Enhancement in Drug supply

Control and Prediction of Solid-State of Pharmaceuticals : Experimental and Computational Approaches

This thesis investigates a number experimental and computational techniques for the invention of stable varieties. additionally, we achieve, as readers, a greater realizing of the foremost elements underpinning solid-structure and variety. a big a part of this thesis highlights experimental paintings conducted on structurally very comparable compounds.

Heterocyclic chemistry in drug discovery

Permits researchers to totally discover the capability to find new prescription drugs between heterocyclic compounds Integrating heterocyclic chemistry and drug discovery, this cutting edge textual content allows readers to appreciate how and why those fields move hand in hand within the powerful perform of medicinal chemistry.

Additional info for Bioactive Heterocyclic Compound Classes: Agrochemicals

Example text

Jacobsen, N. K. (1983) Pestic. , 14, 90–97. T. E. P. (1964) Phytopathology, 54, 941–945. J. (1976) Prog. , 20, 347–383. 23. L. and Benfield, P. (1997) CNS Drugs, 7, 410–416. 24. , Carson, 25. 26. 27. 28. 29. 30. 31. 32. 33. 34. W. (1992) J. Agric. , 40, 1083–1085. M. (2005) Exp. Opin. , 6, 2117–2140. -H. (2004) Pest Manag. , 60, 1007–1012. , and Nishiyama, R. (1987) Nippon Noyaku Gakkaishi, 12, 311–325. D. (2002) J. Med. , 45, 2615–2623. Prakash, A. and Jarvis, B. (1999) Drugs, 58, 1137–1164. E.

2008) in The Practice of Medicinal Chemistry (ed. G. Wermuth), Elsevier, Amsterdam, pp. 290–342; (c) Chen, X. and Wang, W. (2003) Ann. Rep. Med. H. (2001) Curr. Opin. Drug Discov. A. J. (1996) Chem. , 96, 3147–3176; (f) Koyanagi, T. and Haga, T. (1995) in Synthesis and Chemistry of Agrochemicals IV, ACS Symposium Series, Vol. R. G. S. Basarab), American Chemical Society, Washington, DC, pp. 15–24. S. (1983) Drugs, 26, 468–502. Calderbank, A. A. (1984) Drug Chem. , 10, 89–106. N. (1986) Drugs, 32, 60–70.

An empirical rule for amine substituents states that the first chlorine is replaced at 0–5 ◦ C, the second at 30–50 ◦ C, and the third at 70–100 ◦ C [8]. Reactions are typically carried out in the presence of HCl scavengers that may be organic or Bioactive Heterocyclic Compound Classes: Agrochemicals, First Edition. Edited by Clemens Lamberth and J¨urgen Dinges. © 2012 Wiley-VCH Verlag GmbH & Co. KGaA. Published 2012 by Wiley-VCH Verlag GmbH & Co. KGaA. 1 1,2,4-Triazine 1,2,3-Triazine Triazine regioisomers.

Download PDF sample

Download Bioactive Heterocyclic Compound Classes: Agrochemicals by Clemens Lamberth, J?rgen Dinges PDF
Rated 4.45 of 5 – based on 49 votes